Eluxadoline may increase the systemic exposure of coadministered OATP1B1 substrates. Monitor Closely (1)eluxadoline increases levels of ursodiol by decreasing metabolism. Monitor Closely (1)crofelemer increases levels of ursodiol by Other (see comment). Minor (1)colestipol decreases effects of ursodiol by pharmacodynamic antagonism. Minor (1)colesevelam decreases effects of ursodiol by pharmacodynamic antagonism. Minor (1)cholestyramine decreases effects of ursodiol by pharmacodynamic antagonism. Monitor Closely (1)calcium carbonate decreases effects of ursodiol by pharmacodynamic antagonism. Monitor Closely (1)aluminum hydroxide decreases effects of ursodiol by pharmacodynamic antagonism. Mestranol decreases effects of ursodiol by pharmacodynamic antagonism. Minor/Significance Unknown.Ĭolestipol decreases effects of ursodiol by pharmacodynamic antagonism. Minor/Significance Unknown.Ĭolesevelam decreases effects of ursodiol by pharmacodynamic antagonism. Use Caution/Monitor.Ĭholestyramine decreases effects of ursodiol by pharmacodynamic antagonism. Sodium citrate/citric acid decreases effects of ursodiol by pharmacodynamic antagonism. Sodium bicarbonate decreases effects of ursodiol by pharmacodynamic antagonism. Eluxadoline may increase the systemic exposure of coadministered OATP1B1 substrates.Įthinylestradiol decreases effects of ursodiol by pharmacodynamic antagonism. Use Caution/Monitor.Ĭomment: Crofelemer has the potential to inhibit transporters MRP2 and OATP1A2 at concentrations expected in the gut unlikely to inhibit systemically because minimally absorbed.Įluxadoline increases levels of ursodiol by decreasing metabolism. ![]() Use Caution/Monitor.Ĭrofelemer increases levels of ursodiol by Other (see comment). Use Caution/Monitor.Ĭalcium carbonate decreases effects of ursodiol by pharmacodynamic antagonism. ![]() Aluminum hydroxide decreases effects of ursodiol by pharmacodynamic antagonism.
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